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ZOTATIFIN

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number2098191-53-6
INCI Name4-[(2S,3R,4S,5S,6R)-4-[(dimethylamino)methyl]-2,3-dihydroxy-10,12-dimethoxy-5-phenyl-7-oxa-11-azatricyclo[6.4.0.02,6]dodeca-1(12),8,10-trien-6-yl]benzonitrile
PubChem CID 129138801
Molecular FormulaC28H29N3O5
InChIKeyInChI=1S/C28H29N3O5/c1-31(2
SMILESCN(C)C[C@@H]1[C@H]([C@]2([C@@]([C@@H]1O)(C3=C(N=C(C=C3O2)OC)OC)O)C4=CC=C(C=C4)C#N)C5=CC=CC=C5
Known Aliases (7)
Common Name
EFT-226 EFT226 zotatifin [INN] ZOTATIFIN [USAN] Zotatifin [WHO-DD]
Scientific Name
4-{(5aR,6S,7S,8R,8aS)-7-[(Dimethylamino)methyl]-8,8a-dihydroxy-1,3-dimethoxy-6-phenyl-6,7,8,8a-tetrahydro-5aH-cyclopenta[4,5]furo[3,2-c]pyridin-5a-yl}benzonitrile BENZONITRILE, 4-((5AR,6S,7S,8R,8AS)-7-((DIMETHYLAMINO)METHYL)-6,7,8,8A-TETRAHYDRO-8,8A-DIHYDROXY-1,3-DIMETHOXY-6-PHENYL-5AH-CYCLOPENTA(4,5)FURO(3,2-C)PYRIDIN-5A-YL)-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) 2EWN8Z05CN ZOTATIFIN CAS: 2098191-53-6
INN: 10998
USAN: HI-68
SMS_ID: 300000005954
PUBCHEM: 129138801
FDA UNII: 2EWN8Z05CN
EPA CompTox: DTXSID001022536
NCI_THESAURUS: C165746
Record Info
ID3ymtdvneWREqrGrZFkUWH6
CreatedApril 10, 2026, 8:28 p.m.
ModifiedApril 11, 2026, 12:33 a.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)