Skip to main content

ZIPALERTINIB

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number1661854-97-2
INCI NameN-[(8S)-4-amino-6-methyl-5-quinolin-3-yl-8,9-dihydropyrimido[5,4-b]indolizin-8-yl]prop-2-enamide
PubChem CID 117918742
Molecular FormulaC23H20N6O
InChIKeyInChI=1S/C23H20N6O/c1-3-18(
SMILESCC1=C[C@@H](CN2C1=C(C3=C(N=CN=C32)N)C4=CC5=CC=CC=C5N=C4)NC(=O)C=C
Known Aliases (10)
Common Name
CLN-081 CLN081 TAS-6417 TAS6417 TPC-064 TPC064 zipalertinib [INN] ZIPALERTINIB [USAN] Zipalertinib [WHO-DD]
Scientific Name
2-PROPENAMIDE, N-((8S)-4-AMINO-8,9-DIHYDRO-6-METHYL-5-(3-QUINOLINYL)PYRIMIDO(5,4-B)INDOLIZIN-8-YL)-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) T4YMU8TW9H ZIPALERTINIB CAS: 1661854-97-2
INN: 11972
USAN: NO-08
SMS_ID: 300000011362
PUBCHEM: 117918742
FDA UNII: T4YMU8TW9H
NCI_THESAURUS: C165567
Record Info
ID4hXv8eRU9bVHKWatvSJZQZ
CreatedApril 10, 2026, 8:54 p.m.
ModifiedApril 10, 2026, 11:04 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)