Skip to main content

ZIBOTENTAN

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number186497-07-4
INCI NameN-(3-methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide
PubChem CID 9910224
Molecular FormulaC19H16N6O4S
InChIKeyInChI=1S/C19H16N6O4S/c1-12-
SMILESCC1=CN=C(C(=N1)OC)NS(=O)(=O)C2=C(N=CC=C2)C3=CC=C(C=C3)C4=NN=CO4
Known Aliases (11)
Common Name
N-(3-METHOXY-5-METHYLPYRAZIN-2-YL)-2-(4-(1,3,4-OXADIAZOL-2-YL)PHENYL)PRIDINE-3-SULFONAMIDE ZD-4054 ZD4054 zibotentan [INN] ZIBOTENTAN [JAN] ZIBOTENTAN [MART.] ZIBOTENTAN [MI] ZIBOTENTAN [USAN] Zibotentan [WHO-DD]
Scientific Name
3-PYRIDINESULFONAMIDE, N-(3-METHOXY-5-METHYL-2-PYRAZINYL)-2-(4-(1,3,4-OXADIAZOL-2-YL)PHENYL)- N-(3-Methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) 8054MM4902 ZIBOTENTAN CAS: 186497-07-4
INN: 8664
MESH: C511404
USAN: UU-90
EVMPD: SUB32097
ChEMBL: CHEMBL1628688
SMS_ID: 100000124399
PUBCHEM: 9910224
FDA UNII: 8054MM4902
DRUG BANK: DB06629
WIKIPEDIA: ZIBOTENTAN
EPA CompTox: DTXSID70870171
MERCK INDEX: m11590
NCI_THESAURUS: C48430
Record Info
ID6NGBQ4HkzZKx9Yn9w4eGjA
CreatedApril 10, 2026, 11:03 p.m.
ModifiedApril 10, 2026, 11:13 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)