Skip to main content

Zelenirstat

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number1215011-08-7
INCI Name2,6-dichloro-N-[1,5-dimethyl-3-(2-methylpropyl)pyrazol-4-yl]-4-(2-piperazin-1-yl-4-pyridinyl)benzenesulfonamide
PubChem CID 58561243
Molecular FormulaC24H30Cl2N6O2S
InChIKeyInChI=1S/C24H30Cl2N6O2S/c1-
SMILESCC1=C(C(=NN1C)CC(C)C)NS(=O)(=O)C2=C(C=C(C=C2Cl)C3=CC(=NC=C3)N4CCNCC4)Cl
Known Aliases (9)
Common Name
CCI-002 DDD-86481 DDD86481 PCLX-001 PCLX 001 [WHO-DD] zelenirstat [INN]
Scientific Name
2,6-Dichloro-N-[1,5-dimethyl-3-(2-methylpropyl)-1H-pyrazol-4-yl]-4-[2-(1-piperazinyl)-4-pyridinyl]benzenesulfonamide 2,6-dichloro-N-[1,5-dimethyl-3-(2-methylpropyl)-1Hpyrazol-4-yl]-4-[2-(piperazin-1-yl)pyridin-4-yl]benzene-1-sulfonamide Benzenesulfonamide, 2,6-dichloro-N-[1,5-dimethyl-3-(2-methylpropyl)-1H-pyrazol-4-yl]-4-[2-(1-piperazinyl)-4-pyridinyl]-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) 5HY8BYC3Q6 Zelenirstat CAS: 1215011-08-7
INN: 12737
SMS_ID: 300000054573
PUBCHEM: 58561243
FDA UNII: 5HY8BYC3Q6
NCI_THESAURUS: C180576
FDA ORPHAN DRUG: 904722
Record Info
ID92FyDLsyvWT7amFW2j3gUN
CreatedApril 10, 2026, 8:46 p.m.
ModifiedApril 10, 2026, 11:03 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)