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Zandatrigine

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number2154406-04-7
INCI Name4-[[(3S)-1-benzylpyrrolidin-3-yl]-methylamino]-2-fluoro-5-methyl-N-(1,3-thiazol-4-yl)benzenesulfonamide
PubChem CID 132141687
Molecular FormulaC22H25FN4O2S2
InChIKeyInChI=1S/C22H25FN4O2S2/c1-1
SMILESCC1=CC(=C(C=C1N(C)[C@H]2CCN(C2)CC3=CC=CC=C3)F)S(=O)(=O)NC4=CSC=N4
Known Aliases (7)
Common Name
NBI-921352 XEN-901 XEN901 zandatrigine [INN] ZANDATRIGINE [USAN]
Scientific Name
4-{[(3S)-1-benzylpyrrolidin-3-yl](methyl)amino}-2-fluoro-5-methyl-N-(1,3-thiazol-4-yl)benzene-1-sulfonamide Benzenesulfonamide, 2-fluoro-5-methyl-4-[methyl[(3S)-1-(phenylmethyl)-3-pyrrolidinyl]amino]-N-4-thiazolyl-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) SV2WPA4R4J Zandatrigine CAS: 2154406-04-7
INN: 12252
USAN: MN-54
SMS_ID: 300000026612
PUBCHEM: 132141687
FDA UNII: SV2WPA4R4J
NCI_THESAURUS: C190486
FDA ORPHAN DRUG: 762220
Record Info
ID9QGh5GSjW5HfBoXpjfNSZC
CreatedApril 10, 2026, 10:03 p.m.
ModifiedApril 10, 2026, 11:35 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)