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Zongertinib

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number2728667-27-2
INCI NameN-[1-[4-[3-methyl-4-(1-methylbenzimidazol-5-yl)oxyanilino]pyrimido[5,4-d]pyrimidin-6-yl]piperidin-4-yl]prop-2-enamide
PubChem CID 160283094
Molecular FormulaC29H29N9O2
InChIKeyInChI=1S/C29H29N9O2/c1-4-26
SMILESCC1=C(C=CC(=C1)NC2=NC=NC3=CN=C(N=C32)N4CCC(CC4)NC(=O)C=C)OC5=CC6=C(C=C5)N(C=N6)C
Known Aliases (7)
Common Name
BI-1810631 BI1810631 zongertinib [INN] ZONGERTINIB [USAN] Zongertinib [WHO-DD]
Scientific Name
2-Propenamide, N-[1-[8-[[3-methyl-4-[(1-methyl-1H-benzimidazol-5-yl)oxy]phenyl]amino]pyrimido[5,4-d]pyrimidin-2-yl]-4-piperidinyl]- N-[1-(8-{3-methyl-4-[(1-methyl-1H-1,3-benzimidazol-5- yl)oxy]anilino}pyrimido[5,4-d]pyrimidin-2-yl)piperidin-4- yl]prop-2-enamide
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) DRH7R67UVL Zongertinib CAS: 2728667-27-2
INN: 12474
USAN: MN-24
SMS_ID: 300000031413
PUBCHEM: 160283094
FDA UNII: DRH7R67UVL
NCI_THESAURUS: C199022
Record Info
IDBBBNwMhz3hghYmGHLwySY3
CreatedApril 10, 2026, 8:30 p.m.
ModifiedApril 11, 2026, 12:34 a.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)