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Zagociguat

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number2201048-82-8
INCI Name8-[(2-fluorophenyl)methyl]-6-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]imidazo[1,2-a]pyrazine
PubChem CID 134304734
Molecular FormulaC16H10F4N6
InChIKeyInChI=1S/C16H10F4N6/c17-10-
SMILESC1=CC=C(C(=C1)CC2=NC(=CN3C2=NC=C3)C4=NNC(=N4)C(F)(F)F)F
Known Aliases (7)
Common Name
8-[(2-fluorophenyl)methyl]-6-[5-(trifluoromethyl)-4H-1,2,4-triazol-3-yl]imidazo[1,2-a]pyrazine CY-6463 CY6463 IW-6463 zagociguat [INN] ZAGOCIGUAT [USAN]
Scientific Name
Imidazo[1,2-a]pyrazine, 8-[(2-fluorophenyl)methyl]-6-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) H7KEN3O8AI Zagociguat CAS: 2201048-82-8
INN: 11923
USAN: LM-15
SMS_ID: 300000000580
PUBCHEM: 134304734
FDA UNII: H7KEN3O8AI
NCI_THESAURUS: C188581
FDA ORPHAN DRUG: 931423
Record Info
IDGcKQ2khvQTyau5qEV5z6Rz
CreatedApril 10, 2026, 9:01 p.m.
ModifiedApril 10, 2026, 11:40 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)