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ZETELETINIB

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number2216753-97-6
INCI Name2-[6-(6,7-dimethoxyquinolin-3-yl)-3-pyridinyl]-N-[3-(1,1,1-trifluoro-2-methylpropan-2-yl)-1,2-oxazol-5-yl]acetamide
PubChem CID 134391533
Molecular FormulaC25H23F3N4O4
InChIKeyInChI=1S/C25H23F3N4O4/c1-24
SMILESCC(C)(C1=NOC(=C1)NC(=O)CC2=CN=C(C=C2)C3=CN=C4C=C(C(=CC4=C3)OC)OC)C(F)(F)F
Known Aliases (10)
Common Name
BOS-172738 BOS172738 CAXM-1190B DS-5010B RET INHIBITOR DS-5010 zeteletinib [INN] ZETELETINIB [USAN] Zeteletinib [WHO-DD]
Scientific Name
2-(6-(6,7-DIMETHOXYQUINOLIN-3-YL)PYRIDINE-3-YL))-N-(3-(1,1,1-TRIFLUORO-2-METHYLPROPAN-2-YL)-1,2-OXAZOL-5-YL)ACETAMIDE 3-PYRIDINEACETAMIDE, 6-(6,7-DIMETHOXY-3-QUINOLINYL)-N-(3-(2,2,2-TRIFLUORO-1,1-DIMETHYLETHYL)-5-ISOXAZOLYL)-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) EP0P7SHM0U ZETELETINIB CAS: 2216753-97-6
INN: 11523
USAN: KL-16
SMS_ID: 300000026761
PUBCHEM: 134391533
FDA UNII: EP0P7SHM0U
NCI_THESAURUS: C158093
Record Info
IDUAa5dz7K37QAgSioBGs57p
CreatedApril 10, 2026, 8:34 p.m.
ModifiedApril 11, 2026, 12:35 a.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)