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ZENARESTAT

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number112733-06-9
INCI Name2-[3-[(4-bromo-2-fluorophenyl)methyl]-7-chloro-2,4-dioxoquinazolin-1-yl]acetic acid
PubChem CID 5724
Molecular FormulaC17H11BrClFN2O4
InChIKeyInChI=1S/C17H11BrClFN2O4/c1
SMILESC1=CC2=C(C=C1Cl)N(C(=O)N(C2=O)CC3=C(C=C(C=C3)Br)F)CC(=O)O
Known Aliases (9)
Common Name
CI-1014 FK-366 FR-74366 zenarestat [INN] ZENARESTAT [JAN] ZENARESTAT [MI] ZENARESTAT [USAN] Zenarestat [WHO-DD]
Scientific Name
3-(4-Bromo-2-fluorobenzyl)-7-chloro-3,4-dihydro-2,4-dioxo-1(2H)-quinazolineacetic acid
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) 180C9PJ8JT ZENARESTAT CAS: 112733-06-9
INN: 6748
USAN: KK-39
EVMPD: SUB00145MIG
ChEMBL: CHEMBL10413
SMS_ID: 100000079393
PUBCHEM: 5724
FDA UNII: 180C9PJ8JT
DRUG BANK: DB02132
WIKIPEDIA: Zenarestat
EPA CompTox: DTXSID0047296
MERCK INDEX: m986
NCI_THESAURUS: C72880
Record Info
IDUbXspfBws6qrmeAdPyfpfb
CreatedApril 10, 2026, 8:51 p.m.
ModifiedApril 10, 2026, 11:10 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)