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Zidesamtinib

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number2739829-00-4
INCI Name(19R)-3-ethyl-16-fluoro-10,19-dimethyl-20-oxa-3,4,9,10,11,23-hexazapentacyclo[19.3.1.02,6.08,12.013,18]pentacosa-1(25),2(6),4,8,11,13(18),14,16,21,23-decaen-22-amine
PubChem CID 166560233
Molecular FormulaC22H22FN7O
InChIKeyInChI=1S/C22H22FN7O/c1-4-30
SMILESCCN1C2=C(CC3=NN(N=C3C4=C(C=C(C=C4)F)[C@H](OC5=C(N=CC2=C5)N)C)C)C=N1
Known Aliases (11)
Common Name
NU-0002362 NU-0002362-009 NU-2362-010 NU-520 NUV-520 NVL-520 zidesamtinib [INN] ZIDESAMTINIB [USAN] Zidesamtinib [WHO-DD]
Scientific Name
(14R)-7-Ethyl-16-fluoro-2,14-dihydro-2,14-dimethyl-7H-8,12-metheno-4H-pyrazolo[3,4-h]-1,2,3-triazolo[4,5-k][2,5]benzoxaazacyclotetradecin-11-amine 7H-8,12-Metheno-4H-pyrazolo[3,4-h]-1,2,3-triazolo[4,5-k][2,5]benzoxaazacyclotetradecin-11-amine, 7-ethyl-16-fluoro-2,14-dihydro-2,14-dimethyl-, (14R)-
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) MX5KQV5XHC Zidesamtinib CAS: 2739829-00-4
INN: 12588
USAN: MN-48
SMS_ID: 300000037140
PUBCHEM: 166560233
FDA UNII: MX5KQV5XHC
NCI_THESAURUS: C185422
Record Info
IDUs3zejkJY6PXNUotmkn5Xu
CreatedApril 10, 2026, 10:21 p.m.
ModifiedApril 10, 2026, 11:39 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)