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XIMELAGATRAN

Chemical FDA Substance Registry (openFDA)
Chemical Identification
CAS Number192939-46-1
INCI Nameethyl 2-[[(1R)-1-cyclohexyl-2-[(2S)-2-[[4-(N'-hydroxycarbamimidoyl)phenyl]methylcarbamoyl]azetidin-1-yl]-2-oxoethyl]amino]acetate
PubChem CID 656635
Molecular FormulaC24H35N5O5
InChIKeyInChI=1S/C24H35N5O5/c1-2-34
SMILESCCOC(=O)CN[C@H](C1CCCCC1)C(=O)N2CC[C@H]2C(=O)NCC3=CC=C(C=C3)C(=NO)N
Known Aliases (12)
Common Name
EXANTA H 376/95 H-376/95 ximelagatran [INN] XIMELAGATRAN [JAN] XIMELAGATRAN [MART.] XIMELAGATRAN [MI] XIMELAGATRAN [USAN] XIMELAGATRAN [VANDF] Ximelagatran [WHO-DD]
Scientific Name
ethyl ((R)-1-cyclohexyl-2-((S)-2-((4-((E)-(2-hydroxyhydrazono)methyl)benzyl)carbamoyl)azetidin-1-yl)-2-oxoethyl)glycinate Glycine, N-[(1R)-1-cyclohexyl-2-[(2S)-2-[[[[4-[(hydroxyamino)iminomethyl]phenyl]methyl]amino]carbonyl]-1-azetidinyl]-2-oxoethyl]-, ethyl ester
Data Sources (1)
Source Source ID Name in Source Properties
FDA Substance Registry (openFDA) 49HFB70472 XIMELAGATRAN CAS: 192939-46-1
INN: 8037
MESH: C426686
USAN: OO-32
CHEBI: 65172
EVMPD: SUB16473MIG
ChEMBL: CHEMBL522038
SMS_ID: 100000089522
PUBCHEM: 656635
WHO-ATC: B01AE05
FDA UNII: 49HFB70472
WHO-VATC: QB01AE05
DRUG BANK: DB04898
WIKIPEDIA: Ximelagatran
EPA CompTox: DTXSID5049075
MERCK INDEX: m11544
DRUG CENTRAL: 2852
NCI_THESAURUS: C263
Record Info
IDWNhkTnZqXNPRw9VFq8uBY8
CreatedApril 10, 2026, 9:17 p.m.
ModifiedApril 10, 2026, 11:02 p.m.
EnrichedApril 11, 2026, 12:09 a.m.
Data SourceFDA Substance Registry (openFDA)